产品基本信息

产品名称：BOC-Asp(OMe)-FMK [Boc-D(OMe)-FMK]

CAS：187389-53-3

储存条件：-15℃避光防潮

保质期：12个月

产品物理化学光谱特性

分子量：263.27

溶剂：DMF

激发波长（nm）：N/A

发射波长（nm）：N/A

产品介绍

FMK肽是有效的，可透过细胞的，不可逆的capase抑制剂。它可用于检测和监测体外和体内应用中的细胞凋亡。BOC-ASP（OMe）-FMK是开发和制备基于FMK的capase抑制剂和探针的关键中间体。基于Asp（OMe）-FMK的半胱天冬酶抑制剂是细胞可渗透的并且不可逆地结合活化的半胱天冬酶以阻断细胞凋亡。作为分子链锯的胱天蛋白酶是细胞凋亡反应的核心组成部分。半胱天冬酶是半胱氨酸蛋白酶，其天冬氨酸残基在其底物中裂解。14种已知的哺乳动物半胱天冬酶中至少有7种在细胞凋亡中起重要作用。金畔生物是AAT Bioquest的中国代理商，为您提供优质的BOC-Asp(OMe)-FMK [Boc-D(OMe)-FMK]。

参考文献

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